Leqembi

E25439

Leqembi is an Alzheimer’s disease drug (lecanemab) that targets amyloid-beta plaques to slow cognitive decline in early-stage patients.


Statements (48)
Predicate Object
instanceOf Alzheimer’s disease drug
drug
monoclonal antibody
administeredTo adult patients
approvedBy U.S. Food and Drug Administration
belongsToTherapeuticArea neurodegenerative diseases
neurology
coDevelopedBy Eisai and Biogen
developedBy Biogen
Eisai
hasATCClass N06DX
hasBiomarkerTarget amyloid-beta protofibrils
hasBrandOwner Eisai
hasCommonAdverseEffect ARIA-E (amyloid-related imaging abnormalities with edema)
ARIA-H (amyloid-related imaging abnormalities with microhemorrhages and hemosiderin deposits)
headache
infusion-related reactions
hasContraindicationNote caution in patients on anticoagulant therapy
hasCoPromotionPartner Biogen
hasCountryOfApproval United States
hasDosageForm solution for intravenous infusion
hasDosingFrequency every two weeks
hasDrugClass anti-amyloid beta monoclonal antibody
hasEffect slows cognitive decline compared with placebo in early Alzheimer’s disease
hasFDAIndicationText treatment of Alzheimer’s disease
hasGenericName lecanemab
hasIndication Alzheimer’s disease
mild cognitive impairment due to Alzheimer’s disease
mild dementia stage of Alzheimer’s disease
hasINN lecanemab
hasKeyClinicalTrial CLARITY AD
Study 201
Study 301
hasMolecularType humanized IgG1 monoclonal antibody
hasRegulatoryPathway FDA traditional approval
hasRegulatoryStatus FDA approved
hasRouteOfAdministration intravenous infusion
hasWarning risk of ARIA
indicatedFor early-stage Alzheimer’s disease
isAdministeredIn hospital or infusion center settings
isFirstInClass first anti-amyloid Alzheimer’s drug with full FDA approval (as of 2023)
isUsedWith MRI monitoring for ARIA
mechanismOfAction binds aggregated soluble and insoluble amyloid-beta
reduces amyloid-beta plaques in the brain
previouslyHadRegulatoryPathway FDA accelerated approval
requires confirmation of amyloid-beta pathology
targets amyloid-beta
amyloid-beta plaques

Referenced by (8)
Subject (surface form when different) Predicate
Biogen
Eisai ("Lecanemab")
Eisai
hasProduct
Eisai ("Lecanemab")
Eisai
developed
Eisai ("Leqembi – Alzheimer’s disease")
developedForIndication
Leqembi ("lecanemab")
hasGenericName
Leqembi ("lecanemab")
hasINN

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