fampridine

E153840

Fampridine is a potassium channel blocker medication primarily used to improve walking in adults with multiple sclerosis.

All labels observed (3)

Label Occurrences
fampridine canonical 2
Ampyra 1
dalfampridine 1

How this entity was disambiguated

Statements (47)

Predicate Object
instanceOf medication
potassium channel blocker
small molecule
actsOn central nervous system
approvedBy Food and Drug Administration
surface form: U.S. Food and Drug Administration
approvedFor improvement of walking in adults with multiple sclerosis
belongsToPharmacologicalGroup other nervous system drugs
contraindicatedIn moderate or severe renal impairment
patients with history of seizures
developedBy Acorda Therapeutics
discoveredAs 4-aminopyridine derivative used as a research tool before clinical use
hasAdverseEffect back pain
balance disorder
dizziness
headache
insomnia
nausea
paresthesia
seizures
urinary tract infection
hasATCCode N07XX07
hasBlackBoxWarning risk of seizures
hasBrandName fampridine self-linksurface differs
surface form: Ampyra

Fampyra
hasChemicalClass pyridine derivative
hasDosageForm extended-release tablet
hasDosingFrequency typically twice daily for extended-release formulation
hasEffect increases walking speed in some patients with multiple sclerosis
hasEliminationRoute renal
hasGenericName fampridine self-link
hasHalfLife approximately 5–6 hours in adults with normal renal function
hasInternationalNonproprietaryName fampridine
hasMechanismOfAction blocks voltage-gated potassium channels
enhances conduction in demyelinated axons
hasMolecularFormula C5H6N2
hasPregnancyCategory use only if potential benefit justifies potential risk
hasRegulatoryStatus prescription-only medicine
hasRisk increased seizure risk at higher than recommended doses
hasRouteOfAdministration oral
hasTargetPopulation adults with multiple sclerosis
hasTherapeuticArea neurology
hasUSAN fampridine self-linksurface differs
surface form: dalfampridine
indicatedFor multiple sclerosis
walking disability in multiple sclerosis
metabolizedBy kidney excretion largely unchanged
notRecommendedFor patients younger than 18 years
usedFor improvement of walking in adults with multiple sclerosis

How these facts were elicited

Referenced by (4)

Full triples — surface form annotated when it differs from this entity's canonical label.

Fampyra hasActiveIngredient fampridine
fampridine hasGenericName fampridine self-link
fampridine hasUSAN fampridine self-linksurface differs
this entity surface form: dalfampridine
fampridine hasBrandName fampridine self-linksurface differs
this entity surface form: Ampyra