isatuximab

E852349

Isatuximab is a monoclonal antibody drug used primarily in the treatment of multiple myeloma by targeting and killing malignant plasma cells.

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Statements (46)

Predicate Object
instanceOf CD38-targeting antibody
anticancer drug
biologic medicinal product
immunoglobulin G1
monoclonal antibody
protein-based drug
actsOnCellType CD38-expressing hematologic tumor cells
malignant plasma cells
administrationSchedule repeated intravenous infusions in 28-day cycles
approvedBy European Medicines Agency NERFINISHED
U.S. Food and Drug Administration NERFINISHED
ATCCode L01FX09
bindsTo CD38 antigen on plasma cells
commonAdverseEffect anemia
diarrhea
fatigue
infusion-related reaction
neutropenia
pneumonia
thrombocytopenia
upper respiratory tract infection
developer Sanofi NERFINISHED
drugClass antineoplastic agent
immunomodulating agent
monoclonal antibodies against CD38
EMAAuthorizationYear 2020
FDAApprovalYear 2020
hasINN isatuximab
hasTradeName Sarclisa NERFINISHED
indication multiple myeloma
refractory multiple myeloma
relapsed multiple myeloma
marketingAuthorizationHolder Sanofi NERFINISHED
mechanismOfAction induces antibody-dependent cellular cytotoxicity
induces antibody-dependent cellular phagocytosis
induces complement-dependent cytotoxicity
induces direct apoptosis of tumor cells
molecularType recombinant monoclonal antibody
routeOfAdministration intravenous infusion
targetLocation cell surface of plasma cells
targets CD38 NERFINISHED
therapeuticArea hematologic malignancies
oncology
usedWith carfilzomib
dexamethasone NERFINISHED
pomalidomide

Referenced by (1)

Full triples — surface form annotated when it differs from this entity's canonical label.

CD38 targetOf isatuximab