avelumab

E822413

Avelumab is a human monoclonal antibody immunotherapy drug used to treat certain cancers by blocking the PD-L1 immune checkpoint pathway.

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Statements (48)

Predicate Object
instanceOf antineoplastic agent
immunotherapy drug
monoclonal antibody
administrationSetting healthcare facility
antibodyType IgG1
belongsTo checkpoint inhibitor therapies
bindsTo programmed death-ligand 1 NERFINISHED
combinationIndication first-line treatment of advanced renal cell carcinoma with axitinib
commonAdverseEffect diarrhea
fatigue
infusion-related reactions
nausea
rash
contraindicationCaution severe immune-mediated toxicity history
developedBy Merck KGaA NERFINISHED
Pfizer NERFINISHED
dosingSchedule every 2 weeks in many indications
firstFDAApprovalYear 2017
hasATCCode L01FF03
hasGenericName avelumab NERFINISHED
hasHalfLifeApprox 6 days to 7 days
hasTradeName Bavencio NERFINISHED
immuneRelatedAdverseEffect colitis
endocrinopathies
hepatitis
pneumonitis
indicationRegion European Union NERFINISHED
United States NERFINISHED
indicationType oncology
isFullyHuman true
isHuman true
isPrescriptionOnly true
isRecombinant true
mechanismOfAction blocks PD-1/PD-L1 interaction
enhances T-cell mediated immune response against tumor cells
pharmacologicClass PD-L1 blocking antibody
regulatoryApproval EMA-approved
FDA-approved
requiresMonitoringFor immune-mediated adverse reactions
routeOfAdministration intravenous infusion
targets PD-L1 NERFINISHED
treats locally advanced Merkel cell carcinoma
locally advanced renal cell carcinoma
locally advanced urothelial carcinoma
metastatic Merkel cell carcinoma
metastatic renal cell carcinoma
metastatic urothelial carcinoma
usedInCombinationWith axitinib

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