Onpattro

E446845

Onpattro is an RNA interference (RNAi) therapeutic used to treat polyneuropathy in adults with hereditary transthyretin-mediated (hATTR) amyloidosis.

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Statements (49)

Predicate Object
instanceOf RNA interference therapeutic
drug
orphan drug
prescription medicine
small interfering RNA
actsOn transthyretin mRNA
approvedBy European Medicines Agency NERFINISHED
U.S. Food and Drug Administration NERFINISHED
commonAdverseEffect back pain
fatigue
flushing
headache
infusion-related reaction
nausea
containsExcipient DLin-MC3-DMA
PEGylated lipid
cholesterol
lipid excipients
countryOfFirstApproval United States of America NERFINISHED
developedBy Alnylam Pharmaceuticals NERFINISHED
dosageForm concentrate for solution for infusion
dosingInterval once every three weeks
hasActiveIngredient patisiran NERFINISHED
hasApprovalYear 2018
hasATCCode N07XX13
hasDrugClass gene-silencing therapy
transthyretin expression inhibitor
hasIndication polyneuropathy in adults with hereditary transthyretin-mediated amyloidosis
hasInternationalNonproprietaryName patisiran NERFINISHED
hasLegalStatus prescription only
hasPregnancyCategory not recommended during pregnancy unless clearly needed
hasTherapeuticArea neurology
rare diseases
improves neuropathy impairment scores in hATTR patients
isAdministeredBy healthcare professional
isFormulatedAs lipid nanoparticle
marketingAuthorizationHolder Alnylam Pharmaceuticals NERFINISHED
mayCause vitamin A deficiency
mechanismOfAction RNA interference
silencing of transthyretin gene expression in the liver
reduces serum transthyretin levels
reducesLevelOf transthyretin protein
requires premedication to reduce infusion-related reactions
requiresMonitoringOf vitamin A levels
requiresSupplementationOf vitamin A
routeOfAdministration intravenous infusion
targetOrgan liver
treats hATTR amyloidosis with polyneuropathy
hereditary transthyretin-mediated amyloidosis

Referenced by (1)

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