GABA

E675120

GABA (gamma-aminobutyric acid) is the primary inhibitory neurotransmitter in the mammalian central nervous system, crucial for reducing neuronal excitability and regulating muscle tone and anxiety.

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Statements (51)

Predicate Object
instanceOf gamma-aminobutyric acid
inhibitory neurotransmitter
neurotransmitter
non-proteinogenic amino acid
organic compound
actsIn brain
central nervous system
spinal cord
bindsTo GABA-A receptor NERFINISHED
GABA-B receptor NERFINISHED
GABA-C receptor NERFINISHED
chemicalFormula C4H9NO2
effectViaGABAA hyperpolarizes postsynaptic membrane
increases chloride ion influx
effectViaGABAB activates G-protein-coupled signaling
inhibits calcium channels
opens potassium channels
hasFunctionalGroup amino group
carboxylic acid group
hasIUPACName 4-aminobutanoic acid
hasRole anxiolytic modulator
neuromodulator
primary inhibitory neurotransmitter in the mammalian central nervous system
regulator of muscle tone
regulator of neuronal excitability
isAssociatedWithDisorder Huntington disease NERFINISHED
anxiety disorders
epilepsy
insomnia
isClearedFromSynapseBy GABA transporters
isMetabolizedBy GABA transaminase
isPrimaryInhibitoryNeurotransmitterIn mammalian central nervous system
isReleasedAt chemical synapses
isReleasedBy GABAergic neurons
isReleasedInResponseTo nerve impulse
isStoredIn synaptic vesicles
isSynthesizedByEnzyme glutamate decarboxylase
isSynthesizedFrom glutamate
isTargetOfDrugClass barbiturates
gabapentinoids
isTargetOfDrugClass benzodiazepines
general anesthetics
some anticonvulsants
overallEffectOnNeuron reduces neuronal excitability
receptorTypeInteractedWith ionotropic receptor
metabotropic receptor
regulatesProcess anxiety
muscle tone
seizure threshold
sleep
requiresCofactorForSynthesis pyridoxal phosphate

Referenced by (1)

Full triples — surface form annotated when it differs from this entity's canonical label.

Area X neurotransmitter GABA